JP-2022511496-A5 -

Dates

Publication Date

20221214

Application Date

20191205

Description

In chemical formula 1, A1 is NH or N- C1-2 alkyl, A2 is H, a linear or branched C1-5 alkyl, or a phenyl. X is a substituent selected from the group consisting of -H, halogen, -NO2 , -CN, -SR1 , unsubstituted or C1-10 linear or branched alkyl, unsubstituted or C1-10 linear or branched alkoxy, unsubstituted or C1-10 linear or branched alkoxy, unsubstituted or C6-10 aryl , and unsubstituted or C6-10 aryloxy. Y is a substituent selected from the group consisting of unsubstituted or halogen-substituted C1-10 linear or branched alkyl groups, unsubstituted or halogen-substituted C3-10 cycloalkyl groups, 6-10 membered heterocycloalkyl groups containing unsubstituted or halogen-substituted O or S heteroatoms, unsubstituted or halogen-substituted C1-10 linear or branched alkoxy groups, unsubstituted or halogen - substituted C6-10 aryl groups, and unsubstituted or halogen - substituted C6-10 aryloxy groups. R1 is one or more substituents selected from the group consisting of unsubstituted or C1-10 linear or branched alkyl groups substituted with one or more halogens, unsubstituted or C1-10 linear or branched alkoxy groups substituted with one or more halogens, unsubstituted or C6-10 aryl groups substituted with one or more halogens or C1-10 linear or branched alkyl groups, unsubstituted or C1-2 alkyl- C6-10 aryl groups substituted with one or more halogens or C1-10 linear or branched alkyl groups, and unsubstituted or C6-10 aryloxy groups substituted with one or more halogens or C1-10 linear or branched alkyl groups. In one embodiment of the present invention, preferably, among the substituents of the above chemical formula 1, A1 is NH or N- C1-2 alkyl, A2 is H, a linear or branched C1-5 alkyl, or a phenyl. X is a substituent selected from the group consisting of -H, halogens, -NO2 , -CN, -SR1 , unsubstituted or C1-5 linear or branched alkyls substituted with one or more halogens, unsubstituted or C1-5 linear or branched alkoxys, and phenyls that are unsubstituted or substituted with one or more halogens or C1-10 linear or branched alkyls. Y is a substituent selected from the group consisting of unsubstituted or halogen-substituted C1-6 linear or branched alkyl groups, unsubstituted or halogen-substituted C3-6 cycloalkyl groups, 6-8 atomic heterocycloalkyl groups containing an unsubstituted or halogen-substituted O or S heteroatom, unsubstituted or halogen-substituted C1-6 linear or branched alkoxy groups, unsubstituted or halogen -substituted C6-10 aryl groups, and unsubstituted or halogen -substituted C6-10 aryloxy groups. R1 is selected from the group consisting of unsubstituted or C1-6 linear or branched alkyl groups substituted with one or more halogens, unsubstituted or C1-6 linear or branched alkoxy groups substituted with one or more halogens, unsubstituted or C6-10 aryl groups substituted with one or more halogens or C1-10 linear or branched alkyl groups, and unsubstituted or C6-10 aryloxy groups substituted with one or more halogens or C1-10 linear or branched alkyl groups. In the above reaction formula 3, Y is as defined in the above chemical formula 1, R2 is one or more substituents selected from the group consisting of halogens, unsubstituted or C1-10 linear or branched alkyls with one or more halogens, unsubstituted or C1-10 linear or branched alkoxys with one or more halogens, unsubstituted or substituted C6-10 aryls, and unsubstituted or substituted C6-10 aryloxys, where R3 is independently a C1-10 linear or branched alkyl. In the above reaction formula 5, R3 is one or more substituents selected from the group consisting of halogens, unsubstituted or C1-10 linear or branched alkyls with one or more halogens, unsubstituted or C1-10 linear or branched alkoxys with one or more halogens, unsubstituted or substituted C6-10 aryls, and unsubstituted or substituted C6-10 aryloxys, where R3 is independently a C1-10 linear or branched alkyl.