3-PHENYLPROPYLAMINE DERIVATIVE

Inventors

Кагедзи, Хидеаки
КУКИ, Наоки
ХАЯСИ, Нориюки
МАЦУФУДЗИ, Тецуйоси
АСАХИ, Такаси
БАНДЗО, Саки
ЦУЦУМИ, Синдзи
СИМОНАГА, Марико
ИГАРАСИ, Такуя
ЦУКАДА, Томохару
ЦУДЗИ, Такаси
ФУДЗИИ, Масая
СУГИМОТО, Юуити
ЦУТИЯ, Юто
МУРАКАМИ, Кейго
ИНОУЕ, Хидеказу
ЕБИСАВА, Масаюки

Assignees

ДАЙИТИ САНКИО КОМПАНИ, ЛИМИТЕД

Dates

Publication Date: 20260505
Application Date: 20240927
Priority Date: 20230929

Claims (20)

1. A compound represented by the following formula (1):
[Chem. 1]
Where
A represents -O-, -S-, -NR a - or -CR b R c -,
Where
R a represents hydrogen or C 1-3 alkyl,
R b and R c each independently represent hydrogen, halogen, or C 1-3 alkyl, and
alkyl is unsubstituted or substituted by 1-3 halogens,
each R 1 in n quantities is independently halogen, hydroxy, -CN, C 1-6 alkyl, C 2-6 alkenyl, -OC 1-6 alkyl, -N(H)-C 1-3 alkyl, -N(C 1-3 alkyl) 2 , C 3-7 cycloalkyl or 3-7-membered heterocycloalkyl,
Where
alkyl and alkenyl are each independently unsubstituted or substituted by 1 to 3 halogens,
cycloalkyl and heterocycloalkyl are each independently unsubstituted or substituted with 1-3 groups selected from the group consisting of halogen, unsubstituted C 1-3 alkyl and C 1-3 haloalkyl, and
heterocycloalkyl has 1 or 2 heteroatoms selected from oxygen, nitrogen and sulfur as ring member atoms,
R 2 and R 3 each independently represent hydrogen, halogen, C 1-6 alkyl or C 2-6 alkenyl,
Where
alkyl and alkenyl are each independently unsubstituted or substituted by 1 to 3 halogens,
R 4 is C 1-6 alkyl, -C(=O)-R d (R d is C 1-6 alkyl, C 2-5 alkenyl, C 3-7 cycloalkyl or 3-7-membered heterocycloalkyl), C 6-12 aryl or 6-12-membered heteroaryl,
Where
C 1-6 alkyl is unsubstituted or substituted with 1-3 halogens, C 3-7 cycloalkyl or 3-7-membered heterocycloalkyl,
aryl, heteroaryl, cycloalkyl and heterocycloalkyl are each independently unsubstituted or substituted with 1-3 groups selected from the group consisting of halogen, unsubstituted C 1-3 alkyl and C 1-3 haloalkyl, and